Ufa Woyera wa Rotundine (l-tetrahydropalmatine,l-THP)
Rotundine, yomwe imadziwikanso kuti l-tetrahydropalmatine (l-THP), ndi mankhwala omwe ali ndi mphamvu zochizira matenda zomwe zimakhudza dongosolo la mitsempha ndi dongosolo la mtima. Zanenedwa kuti ili ndi mphamvu zochepetsa ululu, zotonthoza, zopumitsa, komanso zolimbikitsa nkhawa. Kuphatikiza apo, yawonetsedwa kuti ili ndi mphamvu zoteteza kuvulala kwa ubongo ndi myocardial ischemia-reperfusion. Rotundine imadziwikanso chifukwa cha kuthekera kwake kosintha kukana mankhwala ambiri m'maselo a khansa komanso mphamvu zake zoletsa njira za calcium.
Ikhoza kupezeka kuchokera ku tuber ya Stephania tetrandra ndi Corydalis yanhusuo, kapena pogwiritsa ntchito njira zopangira mankhwala. Imapangidwa kuchokera ku tetrahydropalmatine kudzera mu kuchepetsa, kugawanika, ndi alkalization reactions. Tetrahydropalmatine yokhala ndi ayodini imatha kupangidwa kuchokera ku tetrahydropalmatine kudzera mu alkalization ndi oxidation kuti ipangidwenso mobwerezabwereza.
Pa pharmacokinetics, Rotundine imayamwa bwino ikaperekedwa pakamwa ndipo imafalikira makamaka mu minofu ya mafuta, kutsatiridwa ndi mapapo, chiwindi, ndi impso. Imatulutsidwa makamaka kudzera mu impso. Kafukufuku wa makoswe ndi akalulu wasonyeza kuti Rotundine imatha kulowa mu chotchinga cha magazi-ubongo ndikulowa mu minofu ya ubongo, ndi kuchuluka kwa ubongo komwe kumatsika poyerekeza ndi kuchuluka kwa magazi pambuyo pa maola awiri.
Pa zotsatirapo zake zoyipa, Rotundine ingayambitse kugona, chizungulire, kutopa, nseru, komanso nthawi zina kugwedezeka kwa ziwalo. Zosamala zikuphatikizapo kupewa kugwiritsa ntchito kwa amayi apakati ndi oyamwitsa, kudziwa kuthekera kolekerera kugwiritsa ntchito kwa nthawi yayitali, komanso kusamala mukamagwiritsa ntchito limodzi ndi mankhwala ochepetsa nkhawa a mitsempha, komanso kusintha mlingo woyenera ngati pakufunika kutero.
Mwachidule, Rotundine ndi mankhwala okhala ndi zotsatira zosiyanasiyana zamankhwala, ndipo makhalidwe ake amawapangitsa kukhala chinthu chofunikira kwambiri pa kafukufuku wosiyanasiyana, kuphatikizapo kuchepetsa ululu, thanzi la mtima, ndi chithandizo cha khansa. Kuti mudziwe zambiri funsani.grace@biowaycn.com.
Mpumulo wa ululu:Rotundine yawonetsedwa kuti ili ndi mphamvu zochepetsera ululu, zomwe zimapangitsa kuti ikhale yothandiza kuchepetsa ululu ndi kusasangalala.
Zotsatira zotsutsana ndi kutupa:Rotundine yawonetsa mphamvu zotsutsana ndi kutupa, zomwe zingathandize kuchepetsa kutupa ndi zizindikiro zina.
Kupumula ndi kugona tulo:Rotundine yagwiritsidwa ntchito polimbikitsa kupumula ndi kugona, zomwe zimapangitsa kuti ikhale yothandiza pothana ndi nkhawa komanso nkhawa.
Ntchito yoletsa kukalamba kwa maselo:Rotundine yapezeka kuti ikuwonetsa mphamvu zotsutsana ndi ma antioxidants, zomwe zingathandize kuteteza maselo ku kuwonongeka komwe kumachitika chifukwa cha ma free radicals.
Kuthekera kwa chithandizo cha chizolowezi:Kafukufuku wina akusonyeza kuti Rotundine ikhoza kukhala ndi kuthekera kothana ndi vuto la kuledzera komanso zizindikiro zosiya kugwiritsa ntchito mankhwala osokoneza bongo, makamaka kwa anthu omwe amamwa mankhwala osokoneza bongo.
Ubwino wa m'mimba:Rotundine yaphunziridwa kuti ingathandize kuthetsa mavuto a m'mimba, monga kupweteka kwa minofu ndi kusasangalala.
| Kusanthula | Kufotokozera |
| Kuyesa | Tetrahydropalmatine ≥98% |
| Maonekedwe | Ufa wachikasu wopepuka mpaka woyera |
| Phulusa | ≤0.5% |
| Chinyezi | ≤5.0% |
| Mankhwala ophera tizilombo | Zoyipa |
| Zitsulo zolemera | ≤10ppm |
| Pb | ≤2.0ppm |
| As | ≤2.0ppm |
| Fungo | Khalidwe |
| Kukula kwa tinthu | 100% mpaka 80 mauna |
| Zamoyo: | |
| Chiwerengero cha mabakiteriya | ≤1000cfu/g |
| Bowa | ≤100cfu/g |
| Salmgosella | Zoyipa |
| Coli | Zoyipa |
Rotundine imagwira ntchito m'mafakitale angapo, kuphatikizapo:
Makampani Opanga Mankhwala:Rotundine imagwiritsidwa ntchito mumakampani opanga mankhwala chifukwa cha mphamvu zake zochepetsa ululu, kutonthoza, komanso kuletsa nkhawa. Ikhoza kuphatikizidwa mu mankhwala ochepetsa ululu komanso kuchepetsa nkhawa.
Chisamaliro chaumoyo ndi thanzi:Chifukwa cha ubwino wake pa thanzi, Rotundine ingagwiritsidwe ntchito ngati mankhwala othandiza pa thanzi komanso pochiza ululu.
Kafukufuku ndi Chitukuko:Rotundine ili ndi chidwi ndi kafukufuku ndi chitukuko chomwe chimayang'ana kwambiri thanzi la mtima, chithandizo cha khansa, ndi matenda amitsempha chifukwa cha zotsatira zake pa machitidwe awa.
Zakudya zopatsa thanzi:Pali kuthekera kophatikiza Rotundine mu zakudya zopatsa thanzi zomwe zimapangidwa kuti zithandize thanzi labwino.
Ndikofunika kuzindikira kuti kugwiritsa ntchito Rotundine kumatha kusiyana malinga ndi zilolezo za malamulo ndi kafukufuku wopitilira mu makampani onse.
Zogulitsa zathu zimapangidwa pogwiritsa ntchito njira zowongolera khalidwe ndipo zimatsatira miyezo yapamwamba ya njira zopangira. Timaika patsogolo chitetezo ndi khalidwe la malonda athu, ndikuonetsetsa kuti akukwaniritsa zofunikira za malamulo ndi ziphaso zamakampani. Kudzipereka kumeneku ku khalidwe labwino kumafuna kukhazikitsa chidaliro ndi chidaliro pa kudalirika kwa malonda athu. Njira yonse yopangira ndi iyi:
Express
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Panyanja
Kupitirira 300kg, Pafupifupi masiku 30
Pakufunika katswiri wopereka chilolezo kuchokera ku doko kupita ku doko
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Pakufunika katswiri wopereka chithandizo kuchokera ku eyapoti kupita ku eyapoti
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