Chilengedwe cha Campotecin ufa (CPT)

Dzina lina la chinthu:Camptothecaca acumiyata kutulutsa
Botani:Camptothecaca acomata
Ntchito Gawo:Nati / mbewu
Kulingana:98% camptothecin
Maonekedwe:Kuwala kowoneka bwino ufa
Pas ayi.:7689-03-4-4
Njira Yoyesera:Hplc
Mtundu wa Mtundu:Kuchotsa
Mamolecular formula:C20h16N2O4
Kulemera kwa maselo:348.36
Gawo:Gawo la mankhwala ndi chakudya


Tsatanetsatane wazogulitsa

Zidziwitso Zina

Matamba a malonda

Kuyambitsa Zoyambitsa

Chilengedwe cha campotecin ufa (cpp) ndi gawo limodzi lochokera ku mtengo wa camptooteca la camptooteca, limadziwikanso kuti "mtengo wosangalatsa" kapena "mtengo wamoyo." Ndiwochitika mwachilengedwe alkaloid yomwe yapezeka kuti ili ndi anti-khansa yotsutsa. Camptootecin ndi zochokera pansi pake zaphunziridwa chifukwa chogwiritsa ntchito khansa, monga momwe aperewera zoletsa kukula kwa maselo a khansa chifukwa cha kuwonongeka kwa enzyme yowonongeka kwa ma cell a khansa. Ufa wachilengedwe wa Campotecin akufufuzidwa kuti athe ntchito ngati wothandizira mankhwala a chemotherapy ndipo ndi chidwi cha malonda opangira mankhwala a chitukuko cha anti-khansa. Kuti mumve zambiri musazengereze kulumikizana ndigrace@email.com.

Kutanthauzira (coa)

Dzina lazogulitsa Camptothecin
Dzina la Latin Camptothecaca acumiyata
Dzina lina Camptothecin 98%
Gawo la ntchito Chipatso
Chifanizo 98%
Njira Yoyesera Hplc
Kaonekedwe Wopepuka wachikaso wachikasu ufa
Cas No. 7689/3/4
Mol. Fomyula C20h16N2O4
Mol. Kulemera 348.35
Moyo wa alumali zaka 2

 

Chinthu Kuyesa statande Kuyesa rkusalankhula
Kaonekedwe Pawuda Zikugwirizana
Mtundu Ufa wachikasu Zikugwirizana
Kukula kwa tinthu 100% Pass 80 mesh Zikugwirizana
Fungo Khalidwe Zikugwirizana
Kakomedwe Khalidwe Zikugwirizana
Kutayika pakuyanika ≤5.0% 2.20%
Chotsalira poyatsira ≤0.1% 0.05%
Otsalira acetone ≤0.1% Zikugwirizana
Zotsalira za Ethanol ≤0.5% Zikugwirizana
Makuda ≤10ppm Zikugwirizana
Na ≤0.1% <0.1%
Pb ≤3 ppm Zikugwirizana
Mbale zonse <1000cfu / g Zikugwirizana
Yisiti & nkhungu <100 CFU / g Zikugwirizana
E. Coli Wosavomela Zikugwirizana
Nsomba monomolla Wosavomela Zikugwirizana
Kutsiliza: Zogwirizana ndi USP muyezo

Mawonekedwe a malonda

Camptothecin ndi gawo lofunikira. Zojambula zake zimaphatikizapo:
Kuyera Kokwanira:Zogulitsa za Camptothech nthawi zambiri zimakhala ndi kuyera kokwanira, ndikuonetsetsa kuti kwawo ndi chitetezo cha mankhwala ndi kupanga.
Cholinga cha Anti-Cancer:Camptootecin idaphunzitsidwa kwambiri ndikugwiritsidwa ntchito mu gawo la mankhwala a anti-khansa ndipo ali ndi anti-chotupa. Chifukwa chake, chimodzi mwazinthu zomwe zimapangidwa ndi zomwe zingatheke ndi khansa.
Zoyambitsa Zachilengedwe:Zogulitsa zina za Camptotecin zimachokera ku mbewu zachilengedwe ndipo chifukwa chake ndizoyenera kugwiritsa ntchito popanga zinthu zachilengedwe komanso zachilengedwe.
Gawo la garriocecical:Zogulitsa za Camptothech nthawi zambiri zimakwaniritsa miyezo ya zamasamba ndipo ndi yoyenera kugwiritsidwa ntchito pokonzekera mankhwala opanga mankhwala.
Ntchito Zogwiritsira Ntchito Magwiridwe:Zogulitsa za Camptothecnin zitha kugwiritsidwa ntchito pakufufuza kwa mankhwala ndi chitukuko, kukonzekera kwachilengedwe, zinthu zaumoyo zachilengedwe, ndi minda ina, komanso kukhala ndi mwayi wogwiritsa ntchito.

Tiyenera kudziwa kuti camptoothecin ndi zinthu zake zimafunikira kutsatira malamulo oyenera komanso njira zotetezeka pakugwiritsa ntchito.

Ubwino Waumoyo

Chilengedwe cha campotecin ufa, wokhala ndi chiyero chochepa cha 98%, chimalumikizidwa ndi mapindu angapo omwe angakhale ndi thanzi labwino, kuphatikizapo:
Katundu wa anticancer:Camptothecin imadziwika chifukwa cha kufooka kwake kwamphamvu. Zimalepheretsa ntchito ya enzyme tokoomeat i, yomwe ikukhudzana ndi DNA repfikitala ya DNA ndi magawano, zimapangitsa kuti ikhale yofunika kwambiri mu khansa ndi kafukufuku.
Ntchito ya Antioxidant:Camptothecin imawonetsa katundu wa antioxidant, yomwe ingathandize kuchepetsa kupsinjika kwa oxidaking ndikuthana ndi ma radicals aulere mthupi, zomwe zingapangitse thanzi lathunthu.
Zotsatira za Anti-zotupa:Kafukufuku wina akuwonetsa kuti Camptothecin atha kukhala ndi zotsutsana ndi zotupa, zomwe zingakhale zopindulitsa pakuwongolera zotupa ndi zizindikiro zokhudzana.
Zotsatira zoyipa za neuroprotective:Pali kafukufuku wakuwonetsa kuti Camptothecin itha kukhala ndi mitsempha ya neuroprotective, yomwe ingakhale yogwirizana ndi matenda a mitsempha komanso thanzi la ubongo.
Ndikofunikira kudziwa kuti pomwe pampatactootecin ufa ungapatsidwe phindu laumoyo, kugwiritsa ntchito kwake kuyenera kulingaliridwa mosamala, ndipo ndikofunikira kuti mufufuze ndi akatswiri azaumoyo musanazigwiritse ntchito pazinthu zilizonse zathanzi.

Mapulogalamu

Chilengedwe cha campotecin ufa wokhala ndi mafayilo osachepera 98% ali ndi mapulogalamu osiyanasiyana mu minda ya mankhwala opanga mankhwala, matracethicals, ndi kafukufuku. Mapulogalamu ena mwatsatanetsatane ndi:
Kafukufuku wa Khansa ndi Kukula kwa Mankhwala:Camptothecin imaphunziridwa kwambiri chifukwa cha mankhwala ake anticancer. Ufawo ukhoza kugwiritsidwa ntchito pofufuza labotaries pophunzira khansa ya pacciologle, chitukuko cha mankhwala, komanso kuchuluka kwa mankhwala a anticancer.
Mapangidwe a mankhwalaUfa wachilengedwe ufa umagwiritsidwa ntchito pakukula kwa mankhwala opangira mankhwala, monga jakisoni wa mankhwala, mankhwala am`kamwa, kapena mapangidwe am'mimba pochiza mitundu ina ya khansa.
Zogulitsa za Nytracethical:Ufawo ukhoza kuphatikizidwa ndi mankhwala othandizira, monga zakudya zamankhwala, cholinga chofuna kupereka phindu laumoyo wogwirizana ndi antioxidant ndi anti-kutupa zinthu.
Ntchito Zodzikongoletsera:Camptothecin imatha kugwiritsidwa ntchito popanga zinthu zopanga zokongoletsa, zokhala ndi zolimba kapena zachikhalidwe, chifukwa cha kuntioxidant yake yoyiteteza komanso yoteteza khungu.
Kafukufuku ndi Chitukuko:Ufa wachilengedwe ukhoza kugwiritsidwa ntchito ngati chida chofufuzira zingapo maphunziro osiyanasiyana asayansi okhudzana ndi khansa, mankhwala, komanso umisite mankhwala.
Ndikofunikira kudziwa kuti kugwiritsa ntchito camptothecin mu pulogalamu iliyonse kuyenera kukhala kogwirizana ndi malangizo owongolera komanso kuyang'aniridwa ndi akatswiri oyenerera chifukwa cha pharmacolological katundu.

Zotsatira zoyipa

Chilengedwe cha campotecin ufa, ndi mankhwala ake amphamvu, atha kukhala ndi zotsatira zoyipa, makamaka ngati amagwiritsidwa ntchito molakwika kapena popanda kuyang'aniridwa ndi achipatala. Zotsatira zoyipa zomwe zingaphatikizepo:
Poizoni:Camptothecin imadziwika kuti ili ndi zovuta, makamaka pamlingo wapamwamba. Itha kuyambitsa kuwonongeka kwa maselo wamba limodzi ndi maselo omwe akungodukika, zomwe zimapangitsa kuti zikhale zowawa ziwalo zosiyanasiyana.
Mimba zosokoneza kwambiri:Kulowetsa camptothecin kapena zochokera kumatha kumabweretsa zovuta kwambiri monga nseru, kusanza, kutsegula m'mimba, ndi kupweteka kwam'mimba.
Hemotogical zotsatira:Camptothecin ingakhudze kupanga maselo amwazi, zomwe zimayambitsa mikhalidwe monga anemia, leukopenia, kapena thrombocytopenia.
Kukhuta khungu:Kulumikizana mwachindunji ndi camptothecin kapena mayankho ake kungapangitse khungu kapena khungu lawo siligwirizana mwa anthu ena.
Zotsatira zina:Zotsatira zina zomwe zingakhale zovuta zitha kuphatikizapo tsitsi, kutopa, kufooka, komanso kusanthula.
Ndikofunikira kutsindika kuti kugwiritsa ntchito ufa wachilengedwe uyenera kukhala motsogozedwa ndi akatswiri azaumoyo, makamaka opanga matomical kapena mankhwala ake amphamvu komanso oopsa. Kuphatikiza apo, anthu ayenera kudziwa malangizo oyang'anira komanso kusamala mosamala zokhudzana ndi ntchito ndi ntchito ya camptoothecin ndi zochokera.


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